Assay Detail
Binding
CHEMBL663260
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibitory effect on Coagulation factor Xa (FXa) from bovine plasma
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Tissue | Plasma |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Design of selective thrombin inhibitors based on the (R)-Phe-Pro-Arg sequence.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 8.30 | 8.30 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL81521 | — | — | 1 | 8.30 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL81521 | — | Ki | = | 4.97 | nM | 8.30 |