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Assay Detail

CHEMBL663446

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity against the cannabinoid receptor (expt 1)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Cannabinoid receptor 1 (CHEMBL218)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

Structural requirements for binding of anandamide-type compounds to the brain cannabinoid receptor.
Sheskin T, Hanus L, Slager J, Vogel Z, Mechoulam R.
J Med Chem (1997) 40 : 659 -667
PubMed 9057852 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 1 5.28 5.28

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL139037 1 5.28

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL139037 Ki = 5240.0 nM 5.28