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Assay Detail

CHEMBL665255

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Binding
Inhibitory concentration against Pneumocystis carinii Dihydrofolate reductase
10
Total Activities
10
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Pneumocystis carinii
Confidence 9 — Direct single protein target
Curated By Intermediate

Target

Dihydrofolate reductase (CHEMBL1926)
Type SINGLE PROTEIN
Organism Pneumocystis carinii

Publication

Synthesis and biological activities of conformationally restricted, tricyclic nonclassical antifolates as inhibitors of dihydrofolate reductases.
Gangjee A, Shi J, Queener SF.
J Med Chem (1997) 40 : 1930 -1936
PubMed 9191971 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 10 6.39 7.88

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL50514 1 7.88
CHEMBL7492 PIRITREXIM 2.0 1 7.51
CHEMBL119 TRIMETREXATE 4.0 1 7.38
CHEMBL299927 1 5.66
CHEMBL57682 1 5.62
CHEMBL293512 1 5.37
CHEMBL58597 1 5.34
CHEMBL60968 1 -
CHEMBL431740 1 -
CHEMBL57637 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL50514 IC50 = 13.2 nM 7.88
CHEMBL7492 PIRITREXIM IC50 = 31.0 nM 7.51
CHEMBL119 TRIMETREXATE IC50 = 42.0 nM 7.38
CHEMBL299927 IC50 = 2200.0 nM 5.66
CHEMBL57682 IC50 = 2400.0 nM 5.62
CHEMBL293512 IC50 = 4280.0 nM 5.37
CHEMBL58597 IC50 = 4600.0 nM 5.34
CHEMBL60968 IC50 > 5000.0 nM -
CHEMBL431740 IC50 > 1000.0 nM -
CHEMBL57637 IC50 > 2270.0 nM -