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Assay Detail

CHEMBL665363

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Binding
Inhibition of Dihydrohydrofolate reductase(DHFR) of Mycobacterium avium
13
Total Activities
13
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Mycobacterium avium
Confidence 9 — Direct single protein target
Curated By Expert

Target

Dihydrofolate reductase (CHEMBL5457)
Type SINGLE PROTEIN
Organism Mycobacterium avium

Publication

Further studies on 2,4-diamino-5-(2',5'-disubstituted benzyl)pyrimidines as potent and selective inhibitors of dihydrofolate reductases from three major opportunistic pathogens of AIDS.
Rosowsky A, Forsch RA, Queener SF.
J Med Chem (2003) 46 : 1726 -1736
PubMed 12699390 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 13 7.61 9.21

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL7492 PIRITREXIM 2.0 1 9.21
CHEMBL34823 1 8.36
CHEMBL37520 1 8.24
CHEMBL37334 1 8.11
CHEMBL33921 1 7.80
CHEMBL285279 1 7.46
CHEMBL35437 1 7.44
CHEMBL33922 1 7.39
CHEMBL35080 1 7.24
CHEMBL290806 1 7.22
CHEMBL288350 1 7.05
CHEMBL288647 1 6.92
CHEMBL22 TRIMETHOPRIM 4.0 1 6.52

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL7492 PIRITREXIM IC50 = 0.61 nM 9.21
CHEMBL34823 IC50 = 4.4 nM 8.36
CHEMBL37520 IC50 = 5.8 nM 8.24
CHEMBL37334 IC50 = 7.8 nM 8.11
CHEMBL33921 IC50 = 16.0 nM 7.80
CHEMBL285279 IC50 = 35.0 nM 7.46
CHEMBL35437 IC50 = 36.0 nM 7.44
CHEMBL33922 IC50 = 41.0 nM 7.39
CHEMBL35080 IC50 = 57.0 nM 7.24
CHEMBL290806 IC50 = 60.0 nM 7.22
CHEMBL288350 IC50 = 89.0 nM 7.05
CHEMBL288647 IC50 = 120.0 nM 6.92
CHEMBL22 TRIMETHOPRIM IC50 = 300.0 nM 6.52