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Assay Detail

CHEMBL665908

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Compound was tested for binding affinity towards Cytosolic aminopeptidase
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

Aspartyl aminopeptidase (CHEMBL2761)
Type SINGLE PROTEIN
Organism Homo sapiens

Publication

alpha-Keto amide inhibitors of aminopeptidases.
Ocain TD, Rich DH.
J Med Chem (1992) 35 : 451 -456
PubMed 1738140 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 2 5.27 5.27

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL142010 1 5.27
CHEMBL342867 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL142010 Ki = 5400.0 nM 5.27
CHEMBL342867 Ki > 600000.0 nM -