Assay Detail
Binding
CHEMBL665958
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Inhibitory activity against Cholecystokinin type B receptor
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Target
Gastrin/cholecystokinin type B receptor (CHEMBL298) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
The design of a dipeptide library for screening at peptide receptor sites
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 7.48 | 9.52 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1121 | SINCALIDE | 4.0 | 1 | 9.52 |
| CHEMBL165869 | — | — | 1 | 8.77 |
| CHEMBL32301 | — | — | 1 | 4.16 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1121 | SINCALIDE | Ki | = | 0.3 | nM | 9.52 |
| CHEMBL165869 | — | Ki | = | 1.7 | nM | 8.77 |
| CHEMBL32301 | — | Ki | = | 70000.0 | nM | 4.16 |