Assay Detail
Binding
CHEMBL666576
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibitory activity against rat brain Dipeptidyl aminopeptidase using 10 nM of [3H]Leu-enkephalin as substrate
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
New bidentates as full inhibitors of enkephalin-degrading enzymes: synthesis and analgesic properties.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 8.63 | 8.63 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL16457 | — | — | 1 | 8.63 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL16457 | — | IC50 | = | 2.32 | nM | 8.63 |