Assay Detail
Binding
CHEMBL666578
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Inhibitory activity against Dipeptidyl aminopeptidase using 10 nM of [3H]Leu-enkephalin as substrate
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
New bidentates as full inhibitors of enkephalin-degrading enzymes: synthesis and analgesic properties.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 9.03 | 9.05 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL85320 | KELATORPHAN | — | 1 | 9.05 |
| CHEMBL2079630 | — | — | 1 | 9.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL85320 | KELATORPHAN | Ki | = | 0.9 | nM | 9.05 |
| CHEMBL2079630 | — | Ki | = | 1.0 | nM | 9.00 |