Assay Detail
Binding
CHEMBL668374
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Inhibitory concentration against binding of [3H]spiperone to human D4 dopaminergic receptor
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Homo sapiens |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
D4 dopamine receptor-selective compounds from the Chinese plant Phoebe chekiangensis
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 4.37 | 4.41 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL19331 | — | — | 1 | 4.41 |
| CHEMBL2303762 | — | — | 1 | 4.32 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL19331 | — | IC50 | = | 39200.0 | nM | 4.41 |
| CHEMBL2303762 | — | IC50 | = | 47500.0 | nM | 4.32 |