Assay Detail
Binding
CHEMBL672309
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Binding affinity towards Dopamine receptor D2
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Expert |
Publication
Higher-end serotonin receptors: 5-HT(5), 5-HT(6), and 5-HT(7).
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 4 | 6.88 | 8.15 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL281924 | — | — | 1 | 8.15 |
| CHEMBL281923 | — | — | 1 | 7.15 |
| CHEMBL281048 | — | — | 1 | 6.58 |
| CHEMBL27251 | — | — | 1 | 5.65 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL281924 | — | Ki | = | 7.1 | nM | 8.15 |
| CHEMBL281923 | — | Ki | = | 71.0 | nM | 7.15 |
| CHEMBL281048 | — | Ki | = | 261.0 | nM | 6.58 |
| CHEMBL27251 | — | Ki | = | 2250.0 | nM | 5.65 |