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Assay Detail

CHEMBL674589

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Binding
Tested for binding affinity against dopamine receptor D3
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Autocuration

Target

D(3) dopamine receptor (CHEMBL3138)
Type SINGLE PROTEIN
Organism Rattus norvegicus

Publication

Synthesis and optical resolution of (R)- and (S)-trans-7-Hydroxy-2-[N-propyl-N-(3'-iodo-2'-propenyl)amino]tetralin: a new D3 dopamine receptor ligand.
Chumpradit S, Kung MP, Kung HF.
J Med Chem (1993) 36 : 4308 -4312
PubMed 8277513 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Kd 1 9.17 9.17

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL285755 1 9.17

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL285755 Kd = 0.67 nM 9.17