Assay Detail
Functional
CHEMBL675130
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Effective concentration for Dopamine receptor D3 was determined
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Cercopithecidae |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
N-(omega-(4-(2-methoxyphenyl)piperazin-1-yl)alkyl)carboxamides as dopamine D2 and D3 receptor ligands.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 2 | 8.30 | 8.60 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL129022 | — | — | 1 | 8.60 |
| CHEMBL126725 | — | — | 1 | 8.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL129022 | — | EC50 | = | 2.5 | nM | 8.60 |
| CHEMBL126725 | — | EC50 | = | 10.0 | nM | 8.00 |