Assay Detail
Functional
CHEMBL677837
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Inhibitory activity against mammalian FM3A cell
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Cell Type | FM3A |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
Synthesis of 2-fluoronoraristeromycin and its inhibitory activity against Plasmodium falciparum S-adenosyl-L-homocysteine hydrolase.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 2 | 6.14 | 7.14 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL129014 | NORARISTEROMYCIN | — | 1 | 7.14 |
| CHEMBL129469 | — | — | 1 | 5.14 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL129014 | NORARISTEROMYCIN | EC50 | = | 72.0 | nM | 7.14 |
| CHEMBL129469 | — | EC50 | = | 7200.0 | nM | 5.14 |