Assay Detail
Binding
CHEMBL678694
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Dissociation constant for Fibroblast growth factor 2
17
Total Activities
17
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Expert |
Publication
Validation of molecular docking calculations involving FGF-1 and FGF-2.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 17 | 5.11 | 5.93 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL2303816 | — | — | 1 | 5.93 |
| CHEMBL3144211 | — | — | 1 | 5.26 |
| CHEMBL2093120 | — | — | 1 | 5.20 |
| CHEMBL2029141 | — | — | 1 | 4.88 |
| CHEMBL2303818 | — | — | 1 | 4.79 |
| CHEMBL2303817 | — | — | 1 | 4.57 |
| CHEMBL1160124 | — | — | 1 | - |
| CHEMBL1160119 | — | — | 1 | - |
| CHEMBL1160112 | — | — | 1 | - |
| CHEMBL1160111 | — | — | 1 | - |
| CHEMBL1160123 | — | — | 1 | - |
| CHEMBL2029142 | — | — | 1 | - |
| CHEMBL1160117 | NAPHTHALENE TRISULFONATE | — | 1 | - |
| CHEMBL2303821 | — | — | 1 | - |
| CHEMBL1160122 | — | — | 1 | - |
| CHEMBL2303819 | — | — | 1 | - |
| CHEMBL1160126 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL2303816 | — | Kd | = | 1180.0 | nM | 5.93 |
| CHEMBL3144211 | — | Kd | = | 5500.0 | nM | 5.26 |
| CHEMBL2093120 | — | Kd | = | 6300.0 | nM | 5.20 |
| CHEMBL2029141 | — | Kd | = | 13300.0 | nM | 4.88 |
| CHEMBL2303818 | — | Kd | = | 16200.0 | nM | 4.79 |
| CHEMBL2303817 | — | Kd | = | 26700.0 | nM | 4.57 |
| CHEMBL1160124 | — | Kd | = | 258000.0 | nM | - |
| CHEMBL1160119 | — | Kd | = | 249000.0 | nM | - |
| CHEMBL1160112 | — | Kd | = | 5100000.0 | nM | - |
| CHEMBL1160111 | — | Kd | = | 7500000.0 | nM | - |
| CHEMBL1160123 | — | Kd | = | 17400000.0 | nM | - |
| CHEMBL2029142 | — | Kd | = | 343000.0 | nM | - |
| CHEMBL1160117 | NAPHTHALENE TRISULFONATE | Kd | = | 223000.0 | nM | - |
| CHEMBL2303821 | — | Kd | = | 550000.0 | nM | - |
| CHEMBL1160122 | — | Kd | = | 8020000.0 | nM | - |
| CHEMBL2303819 | — | Kd | = | 155000.0 | nM | - |
| CHEMBL1160126 | — | Kd | = | 375000.0 | nM | - |