Assay Detail
Functional
CHEMBL679663
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Agonist activity against Gamma-aminobutyric acid type C (GABA-C) receptor derived from bovine retinal RNA expressed in Xenopus oocytes
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Bos taurus |
| Cell Type | Oocyte |
| Confidence | 4 — Cell-line / Tissue |
| Curated By | Autocuration |
Publication
GABA-Activated ligand gated ion channels: medicinal chemistry and molecular biology.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Kd | 1 | 6.22 | 6.22 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL33086 | t-4-AMINOCROTONIC ACID (TACA) | — | 1 | 6.22 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL33086 | t-4-AMINOCROTONIC ACID (TACA) | Kd | = | 600.0 | nM | 6.22 |