Assay Detail
Binding
CHEMBL679997
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding affinity against [125 I][4Tyr]-bombesin labeled cloned human GRP(gastrin releasing peptide) receptors stably expressed in CHO cells
20
Total Activities
20
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Cell Type | CHO |
| Confidence | 8 — Homologous single protein target |
| Curated By | Expert |
Publication
PD 165929 the first high affinity non-peptide neuromedin-B (NMB) receptor selective antagonist
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 20 | 8.26 | 9.82 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL437027 | BOMBESIN | 1.0 | 1 | 9.82 |
| CHEMBL269432 | — | — | 1 | 9.15 |
| CHEMBL328591 | — | — | 1 | 5.82 |
| CHEMBL329561 | — | — | 1 | - |
| CHEMBL87090 | — | — | 1 | - |
| CHEMBL89153 | — | — | 1 | - |
| CHEMBL315859 | — | — | 1 | - |
| CHEMBL315660 | — | — | 1 | - |
| CHEMBL312851 | — | — | 1 | - |
| CHEMBL328230 | — | — | 1 | - |
| CHEMBL1907682 | — | — | 1 | - |
| CHEMBL89795 | — | — | 1 | - |
| CHEMBL313114 | — | — | 1 | - |
| CHEMBL88174 | — | — | 1 | - |
| CHEMBL89075 | — | — | 1 | - |
| CHEMBL406037 | — | — | 1 | - |
| CHEMBL313829 | — | — | 1 | - |
| CHEMBL1907865 | — | — | 1 | - |
| CHEMBL86828 | — | — | 1 | - |
| CHEMBL92274 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL437027 | BOMBESIN | Ki | = | 0.15 | nM | 9.82 |
| CHEMBL269432 | — | Ki | = | 0.7 | nM | 9.15 |
| CHEMBL328591 | — | Ki | = | 1500.0 | nM | 5.82 |
| CHEMBL329561 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL87090 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL89153 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL315859 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL315660 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL312851 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL328230 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL1907682 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL89795 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL313114 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL88174 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL89075 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL406037 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL313829 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL1907865 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL86828 | — | Ki | > | 10000.0 | nM | - |
| CHEMBL92274 | — | Ki | > | 10000.0 | nM | - |