Assay Detail
Binding
CHEMBL680339
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibition of [3H]CGP-27492 binding to cat Gamma-aminobutyric acid type B receptor
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Felis catus |
| Confidence | 6 — Multiple protein complex / RNA |
| Curated By | Expert |
Publication
Phosphinic acid analogues of GABA. 1. New potent and selective GABAB agonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 7.16 | 7.54 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL113304 | — | — | 1 | 7.54 |
| CHEMBL113396 | — | — | 1 | 6.78 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL113304 | — | IC50 | = | 29.0 | nM | 7.54 |
| CHEMBL113396 | — | IC50 | = | 166.0 | nM | 6.78 |