Assay Detail
Binding
CHEMBL681089
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Compound was tested for the inhibitory effect against Gamma-amino-N-butyrate transaminase from bacteria
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Bacteria |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Target
4-aminobutyrate aminotransferase, mitochondrial (CHEMBL2044) ↗| Type | SINGLE PROTEIN |
| Organism | Homo sapiens |
Publication
4-Amino-2-(substituted methyl)-2-butenoic acids: substrates and potent inhibitors of gamma-aminobutyric acid aminotransferase.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 5.05 | 5.05 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL353363 | — | — | 1 | 5.05 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL353363 | — | Ki | = | 9000.0 | nM | 5.05 |