Assay Detail
Binding
CHEMBL681264
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Compound was tested for the inhibition of Fucosyltransferase 4 alpha 1,3 at 8.5 uM GDP-fucose
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Synthesis of inhibitors of -1,3-fucosyltransferase
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 5 | 4.70 | 5.30 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL384759 | — | — | 1 | 5.30 |
| CHEMBL2029050 | — | — | 1 | 4.09 |
| CHEMBL2303733 | — | — | 1 | - |
| CHEMBL314772 | DEOXYFUCONOJIRIMYCIN | — | 1 | - |
| CHEMBL2029051 | — | — | 1 | - |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL384759 | — | IC50 | = | 5000.0 | nM | 5.30 |
| CHEMBL2029050 | — | IC50 | = | 81000.0 | nM | 4.09 |
| CHEMBL2303733 | — | IC50 | = | 233000.0 | nM | - |
| CHEMBL314772 | DEOXYFUCONOJIRIMYCIN | IC50 | = | 3500000.0 | nM | - |
| CHEMBL2029051 | — | IC50 | > | 500000.0 | nM | - |