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Assay Detail

CHEMBL683047

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Binding affinity against Gamma-aminobutyric acid A receptor alpha-6-beta-3-gamma-2
55
Total Activities
55
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 6 — Multiple protein complex / RNA
Curated By Autocuration

Target

GABA-A receptor; alpha-6/beta-3/gamma-2 (CHEMBL2095190)
Type PROTEIN COMPLEX
Organism Homo sapiens

Publication

Predictive models for GABAA/benzodiazepine receptor subtypes: studies of quantitative structure-activity relationships for imidazobenzodiazepines at five recombinant GABAA/benzodiazepine receptor subtypes [alphaxbeta3gamma2 (x = 1-3, 5, and 6)] via comparative molecular field analysis.
Huang Q, Liu R, Zhang P, He X, McKernan R, Gan T, Bennett DW, Cook JM.
J Med Chem (1998) 41 : 4130 -4142
PubMed 9767648 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
Ki 55 6.98 8.42

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL6597 Ro-154513 1 8.42
CHEMBL415293 1 8.40
CHEMBL6659 1 8.34
CHEMBL58757 1 8.29
CHEMBL6421 1 8.28
CHEMBL130609 1 8.16
CHEMBL133049 1 8.08
CHEMBL6655 1 8.03
CHEMBL133219 1 7.66
CHEMBL7290 1 7.65
CHEMBL58570 1 7.64
CHEMBL286594 1 7.54
CHEMBL341398 1 7.51
CHEMBL6814 1 7.51
CHEMBL336728 1 7.38
CHEMBL57655 1 7.35
CHEMBL336377 1 7.34
CHEMBL416450 1 7.29
CHEMBL415290 Ro-151310 1 7.26
CHEMBL300840 1 7.23
CHEMBL133112 1 7.21
CHEMBL52030 1 7.08
CHEMBL59181 1 6.94
CHEMBL339165 1 6.93
CHEMBL339163 1 6.90
CHEMBL407 FLUMAZENIL 4.0 1 6.83
CHEMBL134175 1 6.82
CHEMBL6440 1 6.78
CHEMBL58385 1 6.75
CHEMBL130416 1 6.75

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL6597 Ro-154513 Ki = 3.8 nM 8.42
CHEMBL415293 Ki = 4.0 nM 8.40
CHEMBL6659 Ki = 4.6 nM 8.34
CHEMBL58757 Ki = 5.1 nM 8.29
CHEMBL6421 Ki = 5.25 nM 8.28
CHEMBL130609 Ki = 6.89 nM 8.16
CHEMBL133049 Ki = 8.28 nM 8.08
CHEMBL6655 Ki = 9.4 nM 8.03
CHEMBL133219 Ki = 22.0 nM 7.66
CHEMBL7290 Ki = 22.5 nM 7.65
CHEMBL58570 Ki = 22.9 nM 7.64
CHEMBL286594 Ki = 28.8 nM 7.54
CHEMBL341398 Ki = 31.0 nM 7.51
CHEMBL6814 Ki = 30.7 nM 7.51
CHEMBL336728 Ki = 42.0 nM 7.38
CHEMBL57655 Ki = 44.3 nM 7.35
CHEMBL336377 Ki = 46.0 nM 7.34
CHEMBL416450 Ki = 51.5 nM 7.29
CHEMBL415290 Ro-151310 Ki = 54.6 nM 7.26
CHEMBL300840 Ki = 58.6 nM 7.23
CHEMBL133112 Ki = 61.0 nM 7.21
CHEMBL52030 Ki = 83.2 nM 7.08
CHEMBL59181 Ki = 113.7 nM 6.94
CHEMBL339165 Ki = 118.0 nM 6.93
CHEMBL339163 Ki = 126.0 nM 6.90
CHEMBL407 FLUMAZENIL Ki = 148.0 nM 6.83
CHEMBL134175 Ki = 150.0 nM 6.82
CHEMBL6440 Ki = 168.0 nM 6.78
CHEMBL58385 Ki = 176.0 nM 6.75
CHEMBL130416 Ki = 180.0 nM 6.75
CHEMBL340546 Ki = 247.0 nM 6.61
CHEMBL337166 Ki = 266.0 nM 6.58
CHEMBL133705 Ki = 267.0 nM 6.57
CHEMBL336636 Ki = 301.0 nM 6.52
CHEMBL335960 Ki = 301.0 nM 6.52
CHEMBL131977 Ki = 325.0 nM 6.49
CHEMBL335888 Ki = 333.0 nM 6.48
CHEMBL129855 Ki = 340.0 nM 6.47
CHEMBL339172 Ki = 361.0 nM 6.44
CHEMBL45174 Ki = 960.0 nM 6.02
CHEMBL43724 Ki = 2930.0 nM 5.53
CHEMBL43718 Ki = 3648.0 nM 5.44
CHEMBL46957 Ki = 8600.0 nM 5.07
CHEMBL43725 Ki = 29500.0 nM 4.53
CHEMBL47853 Ki = 30160.0 nM 4.52
CHEMBL336133 Ki > 1000.0 nM -
CHEMBL59180 Ki > 100.0 nM -
CHEMBL445856 Ki > 1000.0 nM -
CHEMBL295981 Ki > 300.0 nM -
CHEMBL432104 Ki > 300.0 nM -