Assay Detail
Binding
CHEMBL683667
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Inhibition constant against mammalian glutamate dehydrogenase (GDH)
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Target
Glutamate dehydrogenase 1, mitochondrial (CHEMBL4628) ↗| Type | SINGLE PROTEIN |
| Organism | Bos taurus |
Publication
CNAD: a potent and specific inhibitor of alcohol dehydrogenase.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 2 | 4.89 | 5.47 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1161866 | — | — | 1 | 5.47 |
| CHEMBL1235132 | — | — | 1 | 4.30 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1161866 | — | Ki | = | 3400.0 | nM | 5.47 |
| CHEMBL1235132 | — | Ki | = | 50000.0 | nM | 4.30 |