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Assay Detail

CHEMBL687735

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
The compound was tested for cytotoxic activity against HT-29 cell line(human colon adeno carcinoma)
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type HT-29
Confidence 1 — Organism
Curated By Intermediate

Target

HT-29 (CHEMBL384)
Type CELL-LINE
Organism Homo sapiens

Publication

N4-(omega-Aminoalkyl)-1-[(omega-aminoalkyl)amino]-4- acridinecarboxamides: novel, potent, cytotoxic, and DNA-binding agents.
Antonini I, Polucci P, Kelland LR, Spinelli S, Pescalli N, Martelli S.
J Med Chem (2000) 43 : 4801 -4805
PubMed 11123989 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 6.52 7.03

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL145462 1 7.03
CHEMBL9940 1 6.00

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL145462 IC50 = 94.0 nM 7.03
CHEMBL9940 IC50 = 990.0 nM 6.00