Assay Detail
Functional
CHEMBL687922
Review assay metadata, readout intent, target linkage, and publication context from the same page.
In vivo inhibition of human ERalpha/ERbeta co-expressed in HEK 293 cells; 21/840
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | HEK293 |
| Confidence | 5 — Multiple protein complex / RNA |
| Curated By | Autocuration |
Publication
Estrogen receptor ligands. Part 3: The SAR of dihydrobenzoxathiin SERMs.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 1 | 7.68 | 7.68 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL316132 | — | — | 1 | 7.68 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL316132 | — | IC50 | = | 21.0 | nM | 7.68 |