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Assay Detail

CHEMBL687991

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Compound was tested for antiviral activity against HCMV in viral cytopathic effect (CPE) assay
11
Total Activities
11
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Human betaherpesvirus 5
Confidence 1 — Organism
Curated By Intermediate

Target

Human betaherpesvirus 5 (CHEMBL371)
Type ORGANISM
Organism Human betaherpesvirus 5

Publication

Synthesis and antiviral evaluation of halogenated beta-D- and -L-erythrofuranosylbenzimidazoles.
Gudmundsson KS, Tidwell J, Lippa N, Koszalka GW, van Draanen N, Ptak RG, Drach JC, Townsend LB.
J Med Chem (2000) 43 : 2464 -2472
PubMed 10882374 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 11 6.47 7.30

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL610088 1 7.30
CHEMBL311260 1 7.30
CHEMBL605480 1 7.00
CHEMBL312038 1 7.00
CHEMBL473894 1 6.52
CHEMBL609189 1 6.22
CHEMBL610659 1 6.10
CHEMBL608010 1 6.00
CHEMBL606433 1 5.64
CHEMBL609782 1 5.64
CHEMBL608011 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL610088 IC50 = 50.0 nM 7.30
CHEMBL311260 IC50 = 50.0 nM 7.30
CHEMBL605480 IC50 = 100.0 nM 7.00
CHEMBL312038 IC50 = 100.0 nM 7.00
CHEMBL473894 IC50 = 300.0 nM 6.52
CHEMBL609189 IC50 = 600.0 nM 6.22
CHEMBL610659 IC50 = 800.0 nM 6.10
CHEMBL608010 IC50 = 1000.0 nM 6.00
CHEMBL606433 IC50 = 2300.0 nM 5.64
CHEMBL609782 IC50 = 2300.0 nM 5.64
CHEMBL608011 IC50 > 10000.0 nM -