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Assay Detail

CHEMBL689339

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Functional
Inhibition against Primase by coupled primase-DNA polymerase-I assay with the two subunit recombinant HSV-1 helicase primase
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Human alphaherpesvirus 1
Confidence 8 — Homologous single protein target
Curated By Expert

Target

DNA helicase/primase complex protein (CHEMBL4380)
Type SINGLE PROTEIN
Organism Herpes simplex virus (type 1 / strain 17)

Publication

Inhibition of herpes simplex virus type 1 helicase-primase by (dichloroanilino)purines and -pyrimidines.
Crute JJ, Lehman IR, Gambino J, Yang TF, Medveczky P, Medveczky M, Khan NN, Mulder C, Monroe J, Wright GE.
J Med Chem (1995) 38 : 1820 -1825
PubMed 7752206 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 4.23 4.23

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL51613 1 4.23

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL51613 IC50 = 59000.0 nM 4.23