Assay Detail
Functional
CHEMBL690851
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Activity against H157 non-SCLC cells in culture
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | NCI-H157 |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
Terminally alkylated polyamine analogues as chemotherapeutic agents.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 6.03 | 6.10 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL33387 | — | — | 1 | 6.10 |
| CHEMBL86940 | — | — | 1 | 5.96 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL33387 | — | IC50 | = | 800.0 | nM | 6.10 |
| CHEMBL86940 | — | IC50 | = | 1100.0 | nM | 5.96 |