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Assay Detail

CHEMBL690923

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Concentration which caused 50% loss of the monolayer present around the viral plaques in uM
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Human alphaherpesvirus 1
Confidence 1 — Organism
Curated By Expert

Target

Human alphaherpesvirus 1 (CHEMBL377)
Type ORGANISM
Organism Human alphaherpesvirus 1

Publication

Synthesis and biological evaluation of certain alpha,beta-unsaturated ketones and their corresponding fused pyridines as antiviral and cytotoxic agents.
El-Subbagh HI, Abu-Zaid SM, Mahran MA, Badria FA, Al-Obaid AM.
J Med Chem (2000) 43 : 2915 -2921
PubMed 10956199 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 5 6.34 6.92

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL329723 1 6.92
CHEMBL29711 APHIDICOLIN 1 6.23
CHEMBL100106 1 6.20
CHEMBL98369 1 6.18
CHEMBL99296 1 6.16

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL329723 IC50 = 120.0 nM 6.92
CHEMBL29711 APHIDICOLIN IC50 = 590.0 nM 6.23
CHEMBL100106 IC50 = 630.0 nM 6.20
CHEMBL98369 IC50 = 660.0 nM 6.18
CHEMBL99296 IC50 = 690.0 nM 6.16