Assay Detail
Binding
CHEMBL691443
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Binding constant against histamine H1 receptor (in vivo)
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Cavia porcellus |
| Confidence | 9 — Direct single protein target |
| Curated By | Autocuration |
Publication
Naphthosultam derivatives: a new class of potent and selective 5-HT2 antagonists.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 7.60 | 7.60 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL83894 | FANANSERIN | 2.0 | 1 | 7.60 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL83894 | FANANSERIN | Ki | = | 25.0 | nM | 7.60 |