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Assay Detail

CHEMBL691946

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
In vitro inhibition of HMG-CoA reductase of rat liver
17
Total Activities
15
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Confidence 8 — Homologous single protein target
Curated By Expert

Target

3-hydroxy-3-methylglutaryl-coenzyme A reductase (CHEMBL3247)
Type SINGLE PROTEIN
Organism Rattus norvegicus

Publication

Synthesis and biological activity of new HMG-CoA reductase inhibitors. 2. Derivatives of 7-(1H-pyrrol-3-yl)-substituted-3,5-dihydroxyhept-6(E)-enoic (-heptanoic) acids.
Jendralla H, Baader E, Bartmann W, Beck G, Bergmann A, Granzer E, von Kerekjarto B, Kesseler K, Krause R, Schubert W.
J Med Chem (1990) 33 : 61 -70
PubMed 2153213 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 17 7.68 8.60

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL436037 2 8.60
CHEMBL162125 1 8.52
CHEMBL350103 1 8.22
CHEMBL2110171 1 8.22
CHEMBL162642 1 8.15
CHEMBL503 LOVASTATIN 4.0 1 8.10
CHEMBL348798 2 8.05
CHEMBL159951 1 8.05
CHEMBL2375156 1 7.19
CHEMBL2375155 1 7.16
CHEMBL161829 1 7.16
CHEMBL163277 1 7.00
CHEMBL160102 1 6.93
CHEMBL159103 1 6.60
CHEMBL345375 1 6.48

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL436037 IC50 = 2.5 nM 8.60
CHEMBL162125 IC50 = 3.0 nM 8.52
CHEMBL436037 IC50 = 5.0 nM 8.30
CHEMBL350103 IC50 = 6.0 nM 8.22
CHEMBL2110171 IC50 = 6.0 nM 8.22
CHEMBL162642 IC50 = 7.0 nM 8.15
CHEMBL503 LOVASTATIN IC50 = 8.0 nM 8.10
CHEMBL159951 IC50 = 9.0 nM 8.05
CHEMBL348798 IC50 = 9.0 nM 8.05
CHEMBL348798 IC50 = 18.0 nM 7.75
CHEMBL2375156 IC50 = 65.0 nM 7.19
CHEMBL2375155 IC50 = 69.0 nM 7.16
CHEMBL161829 IC50 = 70.0 nM 7.16
CHEMBL163277 IC50 = 100.0 nM 7.00
CHEMBL160102 IC50 = 117.0 nM 6.93
CHEMBL159103 IC50 = 250.0 nM 6.60
CHEMBL345375 IC50 = 330.0 nM 6.48