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Assay Detail

CHEMBL694005

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Functional
antiviral activity in Human cytomegalovirus by plaque assay (HCMV)
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Human betaherpesvirus 5
Confidence 1 — Organism
Curated By Intermediate

Target

Human betaherpesvirus 5 (CHEMBL371)
Type ORGANISM
Organism Human betaherpesvirus 5

Publication

Synthesis and antiproliferative and antiviral activity of 2'-deoxy-2'-fluoroarabinofuranosyl analogs of the nucleoside antibiotics toyocamycin and sangivamycin.
Krawczyk SH, Nassiri MR, Kucera LS, Kern ER, Ptak RG, Wotring LL, Drach JC, Townsend LB.
J Med Chem (1995) 38 : 4106 -4114
PubMed 7562946 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 7 5.80 7.60

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3143101 1 7.60
CHEMBL3143102 1 6.66
CHEMBL473686 1 6.00
CHEMBL2111874 1 5.50
CHEMBL182 GANCICLOVIR 4.0 1 5.13
CHEMBL2112687 1 4.92
CHEMBL2112691 1 4.80

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3143101 IC50 = 25.0 nM 7.60
CHEMBL3143102 IC50 = 220.0 nM 6.66
CHEMBL473686 IC50 = 1000.0 nM 6.00
CHEMBL2111874 IC50 = 3200.0 nM 5.50
CHEMBL182 GANCICLOVIR IC50 = 7400.0 nM 5.13
CHEMBL2112687 IC50 = 12000.0 nM 4.92
CHEMBL2112691 IC50 = 16000.0 nM 4.80