Assay Detail
Functional
CHEMBL694024
Review assay metadata, readout intent, target linkage, and publication context from the same page.
In vitro effective concentration in normal human dermal fibroblasts
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Confidence | 0 — Uncurated / Unknown |
| Curated By | Autocuration |
Publication
Triterpene and diterpene inhibitors of pyruvate dehydrogenase kinase (PDK).
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 2 | 4.89 | 5.77 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL440684 | — | — | 1 | 5.77 |
| CHEMBL13960 | DICHLOROACETIC ACID | 3.0 | 1 | 4.00 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL440684 | — | EC50 | = | 1700.0 | nM | 5.77 |
| CHEMBL13960 | DICHLOROACETIC ACID | EC50 | = | 100000.0 | nM | 4.00 |