Assay Detail
Functional
CHEMBL694853
Review assay metadata, readout intent, target linkage, and publication context from the same page.
In vitro inhibitory potency against human T-cells Rb efflux
40
Total Activities
39
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | T-cell line |
| Confidence | 1 — Organism |
| Curated By | Expert |
Publication
The SAR of UK-78,282: A novel blocker of human T cell Kv1.3 potassium channels
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 40 | 5.85 | 6.70 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL9685 | — | — | 1 | 6.70 |
| CHEMBL9670 | — | — | 1 | 6.70 |
| CHEMBL416700 | — | — | 1 | 6.70 |
| CHEMBL441587 | — | — | 1 | 6.70 |
| CHEMBL265407 | — | — | 1 | 6.40 |
| CHEMBL9224 | — | — | 1 | 6.40 |
| CHEMBL9653 | — | — | 2 | 6.40 |
| CHEMBL9591 | — | — | 1 | 6.30 |
| CHEMBL9606 | — | — | 1 | 6.30 |
| CHEMBL9741 | — | — | 1 | 6.30 |
| CHEMBL9536 | — | — | 1 | 6.16 |
| CHEMBL9329 | — | — | 1 | 6.16 |
| CHEMBL9475 | — | — | 1 | 6.16 |
| CHEMBL9288 | — | — | 1 | 6.10 |
| CHEMBL9455 | — | — | 1 | 5.96 |
| CHEMBL394525 | — | — | 1 | 5.82 |
| CHEMBL417065 | — | — | 1 | 5.82 |
| CHEMBL9279 | — | — | 1 | 5.68 |
| CHEMBL266820 | — | — | 1 | 5.66 |
| CHEMBL9628 | — | — | 1 | 5.62 |
| CHEMBL9570 | — | — | 1 | 5.58 |
| CHEMBL9505 | — | — | 1 | 5.57 |
| CHEMBL265374 | — | — | 1 | 5.55 |
| CHEMBL9330 | — | — | 1 | 5.54 |
| CHEMBL9727 | — | — | 1 | 5.52 |
| CHEMBL265406 | — | — | 1 | 5.50 |
| CHEMBL441588 | — | — | 1 | 5.47 |
| CHEMBL9551 | — | — | 1 | 5.37 |
| CHEMBL9742 | — | — | 1 | 5.26 |
| CHEMBL273421 | — | — | 1 | 5.25 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL9685 | — | IC50 | = | 200.0 | nM | 6.70 |
| CHEMBL441587 | — | IC50 | = | 200.0 | nM | 6.70 |
| CHEMBL9670 | — | IC50 | = | 200.0 | nM | 6.70 |
| CHEMBL416700 | — | IC50 | = | 200.0 | nM | 6.70 |
| CHEMBL9653 | — | IC50 | = | 400.0 | nM | 6.40 |
| CHEMBL9224 | — | IC50 | = | 400.0 | nM | 6.40 |
| CHEMBL9653 | — | IC50 | = | 400.0 | nM | 6.40 |
| CHEMBL265407 | — | IC50 | = | 400.0 | nM | 6.40 |
| CHEMBL9741 | — | IC50 | = | 500.0 | nM | 6.30 |
| CHEMBL9606 | — | IC50 | = | 500.0 | nM | 6.30 |
| CHEMBL9591 | — | IC50 | = | 500.0 | nM | 6.30 |
| CHEMBL9329 | — | IC50 | = | 700.0 | nM | 6.16 |
| CHEMBL9475 | — | IC50 | = | 700.0 | nM | 6.16 |
| CHEMBL9536 | — | IC50 | = | 700.0 | nM | 6.16 |
| CHEMBL9288 | — | IC50 | = | 800.0 | nM | 6.10 |
| CHEMBL9455 | — | IC50 | = | 1100.0 | nM | 5.96 |
| CHEMBL417065 | — | IC50 | = | 1500.0 | nM | 5.82 |
| CHEMBL394525 | — | IC50 | = | 1500.0 | nM | 5.82 |
| CHEMBL9279 | — | IC50 | = | 2100.0 | nM | 5.68 |
| CHEMBL266820 | — | IC50 | = | 2200.0 | nM | 5.66 |
| CHEMBL9628 | — | IC50 | = | 2400.0 | nM | 5.62 |
| CHEMBL9570 | — | IC50 | = | 2600.0 | nM | 5.58 |
| CHEMBL9505 | — | IC50 | = | 2700.0 | nM | 5.57 |
| CHEMBL265374 | — | IC50 | = | 2800.0 | nM | 5.55 |
| CHEMBL9330 | — | IC50 | = | 2900.0 | nM | 5.54 |
| CHEMBL9727 | — | IC50 | = | 3000.0 | nM | 5.52 |
| CHEMBL265406 | — | IC50 | = | 3200.0 | nM | 5.50 |
| CHEMBL441588 | — | IC50 | = | 3400.0 | nM | 5.47 |
| CHEMBL9551 | — | IC50 | = | 4300.0 | nM | 5.37 |
| CHEMBL9742 | — | IC50 | = | 5500.0 | nM | 5.26 |
| CHEMBL273421 | — | IC50 | = | 5600.0 | nM | 5.25 |
| CHEMBL9303 | — | IC50 | = | 5900.0 | nM | 5.23 |
| CHEMBL275328 | — | IC50 | = | 10800.0 | nM | 4.97 |
| CHEMBL9656 | — | IC50 | = | 14000.0 | nM | 4.85 |
| CHEMBL8963 | — | IC50 | = | 17800.0 | nM | 4.75 |
| CHEMBL264921 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL9557 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL9513 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL266558 | — | IC50 | > | 20000.0 | nM | - |
| CHEMBL7460 | — | IC50 | > | 20000.0 | nM | - |