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Assay Detail

CHEMBL697851

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Functional
Inhibitory concentration against Human Jurkat T cells
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type Tumor Cell line
Confidence 1 — Organism
Curated By Intermediate

Target

Tumor Cell line (CHEMBL613974)
Type CELL-LINE
Organism Homo sapiens

Publication

Conformational and quantitative structure-activity relationship study of cytotoxic 2-arylidenebenzocycloalkanones.
Dimmock JR, Kandepu NM, Nazarali AJ, Kowalchuk TP, Motaganahalli N, Quail JW, Mykytiuk PA, Audette GF, Prasad L, Perjési P, Allen TM, Santos CL, Szydlowski J, De Clercq E, Balzarini J.
J Med Chem (1999) 42 : 1358 -1366
PubMed 10212121 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 5.46 5.46

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL29539 1 5.46

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL29539 IC50 = 3500.0 nM 5.46