Assay Detail
Binding
CHEMBL698511
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibitory activity against Inosine-5'-monophosphate dehydrogenase
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 4 — Cell-line / Tissue |
| Curated By | Autocuration |
Target
Inosine-5'-monophosphate dehydrogenase (IMPDH) (CHEMBL2111369) ↗| Type | PROTEIN FAMILY |
| Organism | Homo sapiens |
Publication
Discovery of novel low molecular weight inhibitors of IMPDH via virtual needle screening.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 6.60 | 6.60 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL1207374 | — | — | 1 | 6.60 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL1207374 | — | Ki | = | 250.0 | nM | 6.60 |