Skip to main content
Free research Free research Free assay review with research home and workspace preview
Quick search ChEMBL 36
Assay Detail

CHEMBL698625

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
In vitro anticellular activity expressed as inhibitory concentration for the growth of human uterine cervix carcinoma HeLa S3 cells for a period of 1 hour
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type HeLa
Confidence 1 — Organism
Curated By Intermediate

Target

HeLa (CHEMBL399)
Type CELL-LINE
Organism Homo sapiens

Publication

Synthesis and antitumor activity of duocarmycin derivatives: A-ring pyrrole compounds bearing cinnamoyl groups.
Nagamura S, Asai A, Amishiro N, Kobayashi E, Gomi K, Saito H.
J Med Chem (1997) 40 : 972 -979
PubMed 9083487 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 8.71 8.89

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL369203 1 8.89
CHEMBL176802 1 8.52

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL369203 IC50 = 1.3 nM 8.89
CHEMBL176802 IC50 = 3.0 nM 8.52