Assay Detail
Functional
CHEMBL699455
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Agonist activity in Ishikawa human endometrial cells
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Homo sapiens |
| Cell Type | Ishikawa |
| Confidence | 1 — Organism |
| Curated By | Expert |
Publication
Bone targeted drugs 2. synthesis of estrogens with hydroxyapatite affinity
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| EC50 | 4 | 6.62 | 10.00 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL9225 | HEXESTROL | 4.0 | 1 | 10.00 |
| CHEMBL266377 | — | — | 1 | 5.96 |
| CHEMBL267891 | — | — | 1 | 5.80 |
| CHEMBL9428 | — | — | 1 | 4.70 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL9225 | HEXESTROL | EC50 | = | 0.1 | nM | 10.00 |
| CHEMBL266377 | — | EC50 | = | 1100.0 | nM | 5.96 |
| CHEMBL267891 | — | EC50 | = | 1600.0 | nM | 5.80 |
| CHEMBL9428 | — | EC50 | = | 20000.0 | nM | 4.70 |