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Assay Detail

CHEMBL700207

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Functional
In vitro inhibitory activity against K562 leukemia cells
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type K562
Confidence 1 — Organism
Curated By Intermediate

Target

K562 (CHEMBL385)
Type CELL-LINE
Organism Homo sapiens

Publication

Mitomycin antitumor compounds. 2. Interaction of transition metal ions with mitomycin C. Solution structure and biological activity of a Pd(2+)-MMC complex.
Fiallo MM, Deydier E, Bracci M, Garnier-Suillerot A, Halvorsen K.
J Med Chem (2003) 46 : 1683 -1689
PubMed 12699386 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 2 8.24 9.00

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL105 MITOMYCIN 4.0 1 9.00
CHEMBL295703 1 7.48

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL105 MITOMYCIN IC50 = 1.0 nM 9.00
CHEMBL295703 IC50 = 33.0 nM 7.48