Assay Detail
Binding
CHEMBL700230
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Binding affinity towards opioid kappa receptor using [3H]U-69593 as radioligand
3
Total Activities
3
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
(+/-)-4-[(N-allyl-cis-3-methyl-4-piperidinyl)phenylamino]-N,N-diethylbenzamide displays selective binding for the delta opioid receptor.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 5.33 | 5.48 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL102497 | — | — | 1 | 5.48 |
| CHEMBL13470 | SNC-80 | — | 1 | 5.45 |
| CHEMBL321092 | — | — | 1 | 5.06 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL102497 | — | Ki | = | 3284.0 | nM | 5.48 |
| CHEMBL13470 | SNC-80 | Ki | = | 3535.0 | nM | 5.45 |
| CHEMBL321092 | — | Ki | = | 8695.0 | nM | 5.06 |