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Assay Detail

CHEMBL702428

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Binding
Compound concentration required to reduce HIV-1 Integrase 3'-processing activity by 50%
26
Total Activities
26
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Binding
Organism Human immunodeficiency virus 1
Confidence 9 — Direct single protein target
Curated By Expert

Target

Human immunodeficiency virus type 1 integrase (CHEMBL3471)
Type SINGLE PROTEIN
Organism Human immunodeficiency virus 1

Publication

Geometrically and conformationally restrained cinnamoyl compounds as inhibitors of HIV-1 integrase: synthesis, biological evaluation, and molecular modeling.
Artico M, Di Santo R, Costi R, Novellino E, Greco G, Massa S, Tramontano E, Marongiu ME, De Montis A, La Colla P.
J Med Chem (1998) 41 : 3948 -3960
PubMed 9767632 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 26 5.79 6.77

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL232801 AMITROLE 1 6.77
CHEMBL130911 1 6.70
CHEMBL340775 1 6.70
CHEMBL419981 1 6.70
CHEMBL129073 1 6.22
CHEMBL129964 1 6.16
CHEMBL339815 1 6.10
CHEMBL129148 1 6.05
CHEMBL276080 1 6.00
CHEMBL341135 1 5.89
CHEMBL129510 1 5.64
CHEMBL83598 1 5.52
CHEMBL128000 BUTEIN 1 4.70
CHEMBL140 CURCUMIN 3.0 1 4.52
CHEMBL340202 1 4.52
CHEMBL128729 1 4.43
CHEMBL129913 1 -
CHEMBL65 CAMPTOTHECIN -1.0 1 -
CHEMBL128748 DIMETHYLCURCUMIN 2.0 1 -
CHEMBL17205 CYCLOVALONE 2.0 1 -
CHEMBL129795 ISOLIQUIRITIGENIN 1 -
CHEMBL105350 BISDEMETHOXYCURCUMIN 1 -
CHEMBL423698 1 -
CHEMBL127028 1 -
CHEMBL129134 1 -
CHEMBL44657 ETOPOSIDE 4.0 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL232801 AMITROLE IC50 = 170.0 nM 6.77
CHEMBL130911 IC50 = 200.0 nM 6.70
CHEMBL340775 IC50 = 200.0 nM 6.70
CHEMBL419981 IC50 = 200.0 nM 6.70
CHEMBL129073 IC50 = 600.0 nM 6.22
CHEMBL129964 IC50 = 700.0 nM 6.16
CHEMBL339815 IC50 = 800.0 nM 6.10
CHEMBL129148 IC50 = 900.0 nM 6.05
CHEMBL276080 IC50 = 1000.0 nM 6.00
CHEMBL341135 IC50 = 1300.0 nM 5.89
CHEMBL129510 IC50 = 2300.0 nM 5.64
CHEMBL83598 IC50 = 3000.0 nM 5.52
CHEMBL128000 BUTEIN IC50 = 20000.0 nM 4.70
CHEMBL140 CURCUMIN IC50 = 30000.0 nM 4.52
CHEMBL340202 IC50 = 30000.0 nM 4.52
CHEMBL128729 IC50 = 37000.0 nM 4.43
CHEMBL129913 IC50 > 100000.0 nM -
CHEMBL65 CAMPTOTHECIN IC50 > 100000.0 nM -
CHEMBL128748 DIMETHYLCURCUMIN IC50 > 100000.0 nM -
CHEMBL17205 CYCLOVALONE IC50 > 100000.0 nM -
CHEMBL129795 ISOLIQUIRITIGENIN IC50 > 100000.0 nM -
CHEMBL105350 BISDEMETHOXYCURCUMIN IC50 > 100000.0 nM -
CHEMBL423698 IC50 > 100000.0 nM -
CHEMBL127028 IC50 > 100000.0 nM -
CHEMBL129134 IC50 > 100000.0 nM -
CHEMBL44657 ETOPOSIDE IC50 > 100000.0 nM -