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Assay Detail

CHEMBL703376

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Concentration required to decrease the growth rate to 50% of control was evaluated by determining their ability to inhibit growth of L1210 cells in vitro.
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Mus musculus
Cell Type L1210
Confidence 1 — Organism
Curated By Intermediate

Target

L1210 (CHEMBL386)
Type CELL-LINE
Organism Mus musculus

Publication

Synthesis, antiproliferative, and antiviral activity of certain 4-aminopyrrolo[2,3-d]pyridazine nucleosides: an entry into a novel series of adenosine analogues.
Meade EA, Wotring LL, Drach JC, Townsend LB.
J Med Chem (1992) 35 : 526 -533
PubMed 1310744 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 4 5.81 7.40

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL267099 TUBERCIDIN 1 7.40
CHEMBL62099 1 5.40
CHEMBL611541 1 4.62
CHEMBL610706 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL267099 TUBERCIDIN IC50 = 40.0 nM 7.40
CHEMBL62099 IC50 = 4000.0 nM 5.40
CHEMBL611541 IC50 = 24000.0 nM 4.62
CHEMBL610706 IC50 > 100000.0 nM -