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Assay Detail

CHEMBL704308

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
The compound was tested for growth inhibitory activity against L1210/0 tumor cell lines
9
Total Activities
9
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Mus musculus
Cell Type L1210
Confidence 1 — Organism
Curated By Intermediate

Target

L1210 (CHEMBL386)
Type CELL-LINE
Organism Mus musculus

Publication

Novel pyrimidine and purine derivatives of L-ascorbic acid: synthesis and biological evaluation.
Raić-Malić S, Hergold-Brundić A, Nagl A, Grdisa M, Pavelić K, De Clercq E, Mintas M.
J Med Chem (1999) 42 : 2673 -2678
PubMed 10411487 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 9 5.17 5.70

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL92041 1 5.70
CHEMBL419504 1 5.39
CHEMBL327570 1 5.29
CHEMBL328116 1 5.12
CHEMBL90871 1 5.12
CHEMBL88616 1 4.94
CHEMBL88434 1 4.91
CHEMBL91024 1 4.89
CHEMBL315331 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL92041 IC50 = 2000.0 nM 5.70
CHEMBL419504 IC50 = 4100.0 nM 5.39
CHEMBL327570 IC50 = 5100.0 nM 5.29
CHEMBL328116 IC50 = 7500.0 nM 5.12
CHEMBL90871 IC50 = 7500.0 nM 5.12
CHEMBL88616 IC50 = 11600.0 nM 4.94
CHEMBL88434 IC50 = 12200.0 nM 4.91
CHEMBL91024 IC50 = 12900.0 nM 4.89
CHEMBL315331 IC50 = 110000.0 nM -