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Assay Detail

CHEMBL705272

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Growth inhibition of L1210 cells was measured in the presence of nine different concentrations: 0,0.03,0.1,0.3,1,3,10,30, and 100 uM after 48 hours
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Mus musculus
Cell Type L1210
Confidence 1 — Organism
Curated By Intermediate

Target

L1210 (CHEMBL386)
Type CELL-LINE
Organism Mus musculus

Publication

Synthesis and evaluation of hydroxylated polyamine analogues as antiproliferatives.
Bergeron RJ, Müller R, Bussenius J, McManis JS, Merriman RL, Smith RE, Yao H, Weimar WR.
J Med Chem (2000) 43 : 224 -235
PubMed 10649978 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 1 4.70 4.70

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL44083 BIS(ETHYL)NORSPERMINE 1 4.70

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL44083 BIS(ETHYL)NORSPERMINE IC50 = 20000.0 nM 4.70