Assay Detail
Binding
CHEMBL706514
Review assay metadata, readout intent, target linkage, and publication context from the same page.
Inhibitory activity against LTA 4 hydrolase in epoxide hydrolase assay
1
Total Activities
1
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Expert |
Publication
Kelatorphan and related analogs: potent and selective inhibitors of leukotriene A4 hydrolase
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 1 | 7.75 | 7.75 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL85320 | KELATORPHAN | — | 1 | 7.75 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL85320 | KELATORPHAN | Ki | = | 18.0 | nM | 7.75 |