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Assay Detail

CHEMBL707768

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
The compound was tested for growth inhibitory activity against MCF-7 tumor cell lines
9
Total Activities
9
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type MCF7
Confidence 1 — Organism
Curated By Intermediate

Target

MCF7 (CHEMBL387)
Type CELL-LINE
Organism Homo sapiens

Publication

Novel pyrimidine and purine derivatives of L-ascorbic acid: synthesis and biological evaluation.
Raić-Malić S, Hergold-Brundić A, Nagl A, Grdisa M, Pavelić K, De Clercq E, Mintas M.
J Med Chem (1999) 42 : 2673 -2678
PubMed 10411487 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 9 4.36 4.70

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL91024 1 4.70
CHEMBL88616 1 4.40
CHEMBL328116 1 4.40
CHEMBL92041 1 4.40
CHEMBL88434 1 4.22
CHEMBL327570 1 4.22
CHEMBL90871 1 4.16
CHEMBL419504 1 -
CHEMBL315331 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL91024 IC50 = 20000.0 nM 4.70
CHEMBL88616 IC50 = 40000.0 nM 4.40
CHEMBL328116 IC50 = 40000.0 nM 4.40
CHEMBL92041 IC50 = 40000.0 nM 4.40
CHEMBL88434 IC50 = 60000.0 nM 4.22
CHEMBL327570 IC50 = 60000.0 nM 4.22
CHEMBL90871 IC50 = 70000.0 nM 4.16
CHEMBL419504 IC50 > 100000.0 nM -
CHEMBL315331 IC50 > 100000.0 nM -