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Assay Detail

CHEMBL708887

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Inhibition of growth of MCF-7 breast cancer cells in culture
7
Total Activities
7
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type MCF7
Confidence 1 — Organism
Curated By Intermediate

Target

MCF7 (CHEMBL387)
Type CELL-LINE
Organism Homo sapiens

Publication

Cyclodextrin-derived diorganyl tellurides as glutathione peroxidase mimics and inhibitors of thioredoxin reductase and cancer cell growth.
McNaughton M, Engman L, Birmingham A, Powis G, Cotgreave IA.
J Med Chem (2004) 47 : 233 -239
PubMed 14695837 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 7 5.31 5.85

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL412348 1 5.85
CHEMBL437864 1 5.80
CHEMBL385299 1 5.34
CHEMBL413290 1 5.22
CHEMBL440625 1 5.00
CHEMBL411553 1 4.99
CHEMBL217200 1 4.98

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL412348 IC50 = 1400.0 nM 5.85
CHEMBL437864 IC50 = 1600.0 nM 5.80
CHEMBL385299 IC50 = 4600.0 nM 5.34
CHEMBL413290 IC50 = 6000.0 nM 5.22
CHEMBL440625 IC50 = 10100.0 nM 5.00
CHEMBL411553 IC50 = 10200.0 nM 4.99
CHEMBL217200 IC50 = 10400.0 nM 4.98