Assay Detail
Functional
CHEMBL708935
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Compound was evaluated for the inhibitory activity of L1210 cells
4
Total Activities
4
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Functional |
| Organism | Mus musculus |
| Cell Type | L1210 |
| Confidence | 1 — Organism |
| Curated By | Intermediate |
Publication
Application of the three-dimensional structures of protein target molecules in structure-based drug design.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 4 | 6.25 | 6.82 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL9671 | — | — | 1 | 6.82 |
| CHEMBL9440 | METESIND | 2.0 | 1 | 6.52 |
| CHEMBL275685 | — | — | 1 | 6.42 |
| CHEMBL9728 | — | — | 1 | 5.22 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL9671 | — | IC50 | = | 150.0 | nM | 6.82 |
| CHEMBL9440 | METESIND | IC50 | = | 300.0 | nM | 6.52 |
| CHEMBL275685 | — | IC50 | = | 380.0 | nM | 6.42 |
| CHEMBL9728 | — | IC50 | = | 6000.0 | nM | 5.22 |