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Assay Detail

CHEMBL711580

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Inhibitory concentration for anti-HCMV activity against AD-169 strain in MRC-5 cells
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Homo sapiens
Cell Type MRC5
Confidence 1 — Organism
Curated By Intermediate

Target

MRC5 (CHEMBL614181)
Type CELL-LINE
Organism Homo sapiens

Publication

Antiviral oligo- and polyribonucleotides containing selected triazolo[2,3-a]purines.
Tutonda MG, Buckheit RW, Agrawal VK, Broom AD.
J Med Chem (1998) 41 : 4958 -4964
PubMed 9836613 · DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 5 5.89 6.82

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL3144270 1 6.82
CHEMBL3144269 1 6.37
CHEMBL182 GANCICLOVIR 4.0 1 5.20
CHEMBL3144268 1 5.17
CHEMBL3144271 1 -

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL3144270 IC50 = 150.0 nM 6.82
CHEMBL3144269 IC50 = 430.0 nM 6.37
CHEMBL182 GANCICLOVIR IC50 = 6300.0 nM 5.20
CHEMBL3144268 IC50 = 6700.0 nM 5.17
CHEMBL3144271 IC50 > 2800.0 nM -