Assay Detail
Binding
CHEMBL734011
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Inhibitory concentration towards in human monoamine oxidase A was measured
2
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Inactivation of purified human recombinant monoamine oxidases A and B by rasagiline and its analogues.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| IC50 | 2 | 5.46 | 6.16 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL887 | RASAGILINE | 4.0 | 1 | 6.16 |
| CHEMBL1235738 | AZILECT | — | 1 | 4.75 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL887 | RASAGILINE | IC50 | = | 700.0 | nM | 6.16 |
| CHEMBL1235738 | AZILECT | IC50 | = | 17700.0 | nM | 4.75 |