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Assay Detail

CHEMBL736575

Review assay metadata, readout intent, target linkage, and publication context from the same page.

Functional
Compound was tested for its antagonistic activity against Moloney leukemia virus (MoLV) replication
5
Total Activities
5
Compounds Tested
1
Activity Types
0
Assay Parameters

Assay Information

Assay Type Functional
Organism Moloney murine leukemia virus
Confidence 1 — Organism
Curated By Intermediate

Target

Moloney murine leukemia virus (CHEMBL613500)
Type ORGANISM
Organism Moloney murine leukemia virus

Publication

Synthesis and biological activity of sulfoximine-modified myristic acid analogues
McDonald IA, Nyce PL, Ku GS, Bowlin TL
Bioorg Med Chem Lett (1993) 3 : 1717 -1722
· DOI

Activity Statistics

Type Count Avg pChEMBL Best pChEMBL
IC50 5 5.06 5.57

Compounds Tested

Compound Name Phase Activities Best pChEMBL
CHEMBL45627 CERULENIN 1 5.57
CHEMBL1627198 1 5.30
CHEMBL1627197 1 5.00
CHEMBL1627268 1 4.82
CHEMBL1627196 1 4.62

Activity Data

Compound Name Type Rel. Value Units pChEMBL
CHEMBL45627 CERULENIN IC50 = 2700.0 nM 5.57
CHEMBL1627198 IC50 = 5000.0 nM 5.30
CHEMBL1627197 IC50 = 10000.0 nM 5.00
CHEMBL1627268 IC50 = 15000.0 nM 4.82
CHEMBL1627196 IC50 = 24000.0 nM 4.62