Assay Detail
Binding
CHEMBL746885
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Inhibitor constant was measured against Muscle phosphorylase b in rabbit
3
Total Activities
2
Compounds Tested
1
Activity Types
0
Assay Parameters
Assay Information
| Assay Type | Binding |
| Organism | Oryctolagus cuniculus |
| Confidence | 8 — Homologous single protein target |
| Curated By | Autocuration |
Publication
Efficient inhibition of muscle and liver glycogen phosphorylases by a new glucopyranosylidene-spiro-thiohydantoin.
Activity Statistics
| Type | Count | Avg pChEMBL | Best pChEMBL |
|---|---|---|---|
| Ki | 3 | 5.34 | 5.38 |
Compounds Tested
| Compound | Name | Phase | Activities | Best pChEMBL |
|---|---|---|---|---|
| CHEMBL3351144 | — | — | 2 | 5.38 |
| CHEMBL489798 | — | — | 1 | 5.29 |
Activity Data
| Compound | Name | Type | Rel. | Value | Units | pChEMBL |
|---|---|---|---|---|---|---|
| CHEMBL3351144 | — | Ki | = | 4200.0 | nM | 5.38 |
| CHEMBL489798 | — | Ki | = | 5100.0 | nM | 5.29 |
| CHEMBL3351144 | — | Ki | = | 105000.0 | nM | - |